TargetMol

(-)-U-50488 hydrochloride

Product Code:
 
TAR-T21830
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T21830-200mg200mg£1,248.00
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Quantity:
TAR-T21830-500mg500mg£2,307.00
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This product comes from: United States.
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Further Information

Bioactivity:
(-)-U-50488 hydrochloride ((-)-Trans-(1S,2S)-U-50488 hydrochloride) is a selective kappa-opioid receptor (KOR) agonist (b>K d =2.2 nM) which is a more selective than u-opioid receptor (MOR) (b>K d =430 nM). (-)-U-50488 hydrochloride is a more active enantiomer than (+) trans-(1R,2R) U-50488 or the (?) trans-racemic mixture U-50488. (-)-U-50488 hydrochloride has a potent and sustained anti- HIV effect in fected blood monocyte-derived macrophages (MDM) [1].
CAS:
114528-79-9
Formula:
C19H27Cl3N2O
Molecular Weight:
405.79
Purity:
0.98
SMILES:
Cl.CN([C@H]1CCCC[C@@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1