TargetMol

RO2959 monohydrochloride

Product Code:
 
TAR-T62940
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T62940-100mg100mg£1,235.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
RO2959 monohydrochloride is a potent, selective inhibitor of CRAC channels (IC50: 402 nM) and a potent blocker of Orai1/Stim1 channel-mediated calcium store entry (SOCE) (IC50: 25 nM). A potent inhibitor of human IL-2 production, effectively blocking T cell receptor-triggered gene expression and T cell functional pathways.
CAS:
2309172-44-7
Molecular Weight:
463.93
Purity:
0.98
SMILES:
Cl.O=C(NC1=NC=C(N=C1)C2=C(C)CCN(C3=NC=C(S3)C)C2)C=4C(F)=CC=CC4F