TargetMol

Thalidomide-Piperazine 5-fluoride

Product Code:
 
TAR-T39696
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T39696-100mg100mgEnquire
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TAR-T39696-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
Thalidomide-Piperazine 5-fluoride is a compound developed by synthesizing an E3 ligase ligand-linker conjugate. It incorporates a cereblon ligand derived from Thalidomide and utilizes a linker commonly employed in PROTAC technology.
CAS:
2222114-22-7
Molecular Weight:
360.34
Purity:
0.98
SMILES:
O=C1NC(=O)C(N2C(=O)C3=CC(F)=C(C=C3C2=O)N4CCNCC4)CC1

References

Hexiang Wang, et al. Degradation of androgen receptor (ar) by conjugation of ar antagonists with e3 ligase ligand and methods of use. WO2021058017A1.