TargetMol

KUNG94

Product Code:
 
TAR-T27756
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T27756-100mg100mgEnquire
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TAR-T27756-500mg500mgEnquire
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Further Information

Bioactivity:
KUNG94 is a potent and selective inhibitor of Glucose regulated protein 94 (Grp94) (IC50 = 8 nM), the endoplasmic reticulum resident of the 90 kDa heat shock protein (Hsp90) family.
CAS:
T27756
Molecular Weight:
363.39
Purity:
0.98
SMILES:
FC1=CC=C(CC2=C(O)C=C(O)C(C(N3CC(C=CC=C4)=C4C3)=O)=C2)C=C1

References

Resorcinol-Based Grp94-Selective Inhibitors Anuj Khandelwal,?,?,? Vincent M. Crowley,?,? and Brian S. J. Blagg*,? ?Department of Medicinal Chemistry, The University of Kansas, 1251 Wescoe Hall Drive, Malott Hall 4070, Lawrence, Kansas
66045, United States ?Warren Family Research Center for Drug Discovery and Development and Department of Chemistry & Biochemistry, University of Notre Dame, 305 McCourtney Hall, Notre Dame, Indiana 46556, United States