TargetMol

Lenalidomide-PEG1-azide

Product Code:
 
TAR-T18067
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T18067-100mg100mgEnquire
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TAR-T18067-500mg500mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
Lenalidomide-PEG1-azide is a E3 ligase lgand-linker conjugate. Lenalidomide-PEG1-azide incorporates the Lenalidomide based cereblon ligand and a linker. Lenalidomide-PEG1-azide can be used to design a PROTAC BRD4 Degrader-2[1].
CAS:
2185795-67-7
Molecular Weight:
386.36
Purity:
0.98
SMILES:
[N-]=[N+]=NCCOCC(=O)NC1=CC=CC=2C(=O)N(CC12)C3C(=O)NC(=O)CC3

References

Zhang F, et al. Discovery of a new class of PROTAC BRD4 degraders based on a dihydroquinazolinone derivative and lenalidomide/pomalidomide. Bioorg Med Chem. 2020 Jan 1;28(1):115228.