TargetMol

cIAP1 Ligand-Linker Conjugates 5

Product Code:
 
TAR-T17893
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T17893-100mg100mgEnquire
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TAR-T17893-500mg500mgEnquire
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Further Information

Bioactivity:
cIAP1 Ligand-Linker Conjugates 5 is a chemical compound consisting of an IAP ligand that targets the E3 ubiquitin ligase, and a PROTAC linker. This compound, cIAP1 Ligand-Linker Conjugates 5, is specifically designed for the development of SNIPERs[1].
CAS:
2113688-20-1
Molecular Weight:
729.93
Purity:
0.98
SMILES:
C([C@@H](NC([C@@H](N(C(OC(C)(C)C)=O)C)C)=O)[C@H]1CCCCC1)(=O)N2[C@@](CCC2)(C3=NC(C(=O)C4=CC(OCCOCCOCCN)=CC=C4)=CS3)[H]

References

Shibata N, et al. Development of Protein Degradation Inducers of Androgen Receptor by Conjugation of Androgen Receptor Ligands and Inhibitor of Apoptosis Protein Ligands. J Med Chem. 2018 Jan 25;61(2):543-575.