TargetMol

CCK2R Ligand-Linker Conjugates 1

Product Code:
 
TAR-T17727
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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TAR-T17727-100mg100mgEnquire
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TAR-T17727-500mg500mgEnquire
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Further Information

Bioactivity:
CCK2R Ligand-Linker Conjugate 1 is a hydrophilic peptide linker that conjugates to the cytotoxic antimicrotubule agents Desacetyl Vinblastine Hydrazide (DAVBH) and Tubulysin B Hydrazide (TubBH) as ligand-linker conjugates[1].
CAS:
1452145-13-9
Molecular Weight:
1607.77
Purity:
0.98
SMILES:
C(C(C(C)(C)C)=O)N1C=2C(N(C[C@@H](NC(NC3=CC(C(NCCCCCCCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(O)=O)CS)=O)CCC(NC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O)=O)=O)CCC(O)=O)=O)CCC(NC[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O)=O)=O)CCC(O)=O)=O)=O)=CC=C3)=O)C1=O)C4CCCCC4)=CC=CC2

References

Wayua C, et al. Selective Tumor Targeting of Desacetyl Vinblastine Hydrazide and Tubulysin B via Conjugation to a Cholecystokinin 2 Receptor (CCK2R) Ligand. Mol Pharm. 2015 Jul 6;12(7):2477-83.