TargetMol

6-Alpha Naloxol

Product Code:
 
TAR-T10180
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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Further Information

Bioactivity:
6-Alpha Naloxol(Alpha-Naloxol) is an opioid antagonist and is a human metabolite of naloxone.
CAS:
20410-95-1
Formula:
C19H23NO4
Molecular Weight:
329.39
Purity:
0.98
SMILES:
O[C@]12[C@@]34C=5C(O[C@]3([C@@H](O)CC1)[H])=C(O)C=CC5C[C@H]2N(CC=C)CC4

References

Weinstein SH, et al. Metabolites of naloxone in human urine. J Pharm Sci. 1971 Oct;60(10):1567-8. Csaba Simon, et al. Stereoselective synthesis of ?-naltrexol, ?-naloxol ?-naloxamine, ?-naltrexamine and related compounds by the application of the mitsunobu reac. Tetrahedron Volume 50, Issue 32, 1994, Pages 9757?9768. Schulteis G, et al. Relative potency of the opioid antagonists naloxone and 6-alpha-naloxol to precipitate withdrawal from acute morphine dependence varies with time post-antagonist. Pharmacol Biochem Behav. 2009 Mar;92(1):157-63.