TargetMol

TM-1

Product Code:
 
TAR-T63012
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T63012-100mg100mgEnquire
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TAR-T63012-50mg50mgEnquire
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TM-1 is a potent pyruvate dehydrogenase kinase (PDHK) inhibitor that inhibits the activity of PDHK1 (IC50: 2.97 uM) and PDHK2 (IC50: 5.2 uM). TM-1 blocks pyruvate dehydrogenase complex (PDHC) phosphorylation and inhibits cancer cell proliferation.
CAS:
921099-13-0
Molecular Weight:
468.55
Purity:
0.98
SMILES:
O=C1OC2=CC(OCCN3CCN(CCO)CC3)=CC=C2C(=C1C=4C=CC(OC)=C(OC)C4)C