TargetMol

PSB-12379

Product Code:
 
TAR-T12569
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T12569-50mg50mgEnquire
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Further Information

Bioactivity:
PSB-12379 is a potent inhibitor of Ecto-5'-Nucleotidase (CD73)(Kis of 9.03 nM (rat) and 2.21 nM (human)).
CAS:
1802226-78-3
Formula:
C18H23N5O9P2
Molecular Weight:
515.35
Purity:
0.98
SMILES:
O[C@H]1[C@](N2C=3C(N=C2)=C(NCC4=CC=CC=C4)N=CN3)(O[C@H](COP(CP(=O)(O)O)(=O)O)[C@H]1O)[H]

References

Bhattarai S, et al. ?,?-Methylene-ADP (AOPCP) Derivatives and Analogues: Development of Potent and Selective ecto-5'-Nucleotidase (CD73) Inhibitors. J Med Chem. 2015 Aug 13;58(15):6248-63.