TargetMol

HDAC-IN-50

Product Code:
 
TAR-T73179
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T73179-5mg5mg£1,010.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T73179-50mg50mg£1,982.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T73179-100mg100mg£2,560.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
HDAC-IN-50 is a potent and orally active FGFR and HDAC dual inhibitor with IC 50 values of 0.18, 1.2, 0.46, 1.4, 1.3, 1.6, 2.6, 13 nM for FGFR1 , FGFR2 , FGFR3 , FGFR4 , HDAC1 , HDAC2 , HDAC6 , HDAC8 , respectively. HDAC-IN-50 induces Apoptosis and cell cycle arrest at G0/G1 phase. HDAC-IN-50 decreases the expression of pFGFR1, pERK , pSTAT3. HDAC-IN-50 shows anti-tumor activity .
CAS:
2653339-26-3
Molecular Weight:
575.7
Purity:
0.98
SMILES:
O=C(NO)CCCCCCN1N=CC(=C1)C2=NC=3C=C(C=CC3N=C2)N(C=4C=C(OC)C=C(OC)C4)CCNC(C)C