TargetMol

CYP1B1-IN-4

Product Code:
 
TAR-T73040
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T73040-5mg5mg£115.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T73040-1mL1 mL * 10 mM (in DMSO)£131.00
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Quantity:
TAR-T73040-10mg10mg£142.00
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Quantity:
TAR-T73040-25mg25mg£213.00
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Quantity:
TAR-T73040-50mg50mg£303.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T73040-100mg100mg£414.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CYP1B1-IN-4 is a selective CYP1B1 inhibitor with an IC50 value of 0.2 nM.CYP1B1-IN-4 is a 2,4-diarylthiazole compound with potential anticancer activity and low cytotoxicity, and is stable in human and rat liver microsomes.
CAS:
2685779-55-7
Molecular Weight:
322.38
Pathway:
Metabolism
Purity:
0.98
SMILES:
N#CC=1C=CC(=CC1)C=2N=C(SC2)C=3C=CC(OC)=CC3OC
Target:
P450

References

Hachey AC, et al. Design of Cytochrome P450 1B1 Inhibitors via a Scaffold-Hopping Approach. J Med Chem. 2023 Jan 12;66(1):398-412.