TargetMol

Theliatinib tartrate

Product Code:
 
TAR-T72431
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T72431-5mg5mg£850.00
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Quantity:
TAR-T72431-50mg50mg£1,661.00
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Quantity:
TAR-T72431-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Theliatinib (Xiliertinib) tartrate is a potent, ATP-competitive, orally active and highly selective EGFR inhibitor with a K i of 0.05 nM and an IC 50 of 3 nM. Theliatinib has an IC 50 of 22 nM for EGFR T790M/L858R mutant . Theliatinib shows >50-fold selectivity for EGFR than other kinases .
CAS:
2413487-72-4
Molecular Weight:
592.6
Purity:
0.98
SMILES:
[C@@H]([C@H](C(O)=O)O)(C(O)=O)O.N(C=1C2=C(C=C(OC)C(NC(=O)N3C[C@]4([C@@](C3)(CCN4C)[H])[H])=C2)N=CN1)C5=CC(C#C)=CC=C5