TargetMol

MPT0G211 mesylate

Product Code:
 
TAR-T61753
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T61753-5mg5mg£850.00
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TAR-T61753-50mg50mg£1,661.00
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Quantity:
TAR-T61753-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
MPT0G211 mesylate is a powerful and selective HDAC6 inhibitor (IC50 = 0.291 nM), with high oral bioavailability. It exhibits remarkable selectivity for HDAC6 over other HDAC isoforms (>1000-fold selectivity). Additionally, MPT0G211 mesylate can effectively cross the blood-brain barrier. In preclinical studies using an Alzheimer's disease model, MPT0G211 mesylate has shown promising results in reducing tau phosphorylation and cognitive deficits. Furthermore, this compound exhibits anti-metastatic and neuroprotective effects, making it a potential candidate for anticancer interventions. [1] [2] [3].
CAS:
2151854-33-8
Formula:
C18H19N3O5S
Molecular Weight:
389.43
Purity:
0.98
SMILES:
CS(O)(=O)=O.ONC(=O)c1ccc(CNc2cccc3cccnc23)cc1