TargetMol

Immunoproteasome inhibitor 1

Product Code:
 
TAR-T61320
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1

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CodeSizePrice
TAR-T61320-5mg5mg£850.00
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Quantity:
TAR-T61320-50mg50mg£1,661.00
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Quantity:
TAR-T61320-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Immunoproteasome inhibitor 1 is a highly potent and reversible inhibitor of both immunoproteasome and proteasome activity. It exhibits time-independent inhibitory effects on immunoproteasome subunits β5c, β1i, and β5i, with respective Ki values of 1.18 uM, 0.27 uM, and 1.91 uM. This compound shows promising potential for the treatment of select neoplastic diseases [1].
CAS:
2755772-63-3
Formula:
C20H26N2O4
Molecular Weight:
358.438
Purity:
0.98
SMILES:
COc1cc2ccn(C\C=C\C(=O)NCCC(C)C)c(=O)c2cc1OC