TargetMol

Helianorphin-19

Product Code:
 
TAR-T41183
Product Group:
 
Peptides
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
 

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CodeSizePrice
TAR-T41183-5mg5mgEnquire
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Further Information

Bioactivity:
Helianorphin-19 is a high affinity, potent and selective κ-opioid receptor (KOR) agonist (Ki = 25 nM; EC50= 45 nM). Helianorphin-19 exhibits approximately 200-fold selectivity for KOR over u and δ-opioid receptors.In vivoHelianorphin-19 shows potent peripheral analgesic efficacy in a mouse model of visceral pain without affecting motor coordination/sedation.
Purity:
0.98

References

Muratspahi? et al (2021) Design of a stable cyclic peptide analgesic derived from sunflower seeds that targets the ?-opioid receptor for the treatment of chronic abdominal pain. J.Med.Chem. 64 9042 PMID: 34162205