TargetMol

P2Y2R/GPR17 antagonist 1

Product Code:
 
TAR-T62420
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T62420-1mg1mg£97.00
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TAR-T62420-5mg5mg£130.00
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TAR-T62420-1mL1 mL * 10 mM (in DMSO)£131.00
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TAR-T62420-10mg10mg£158.00
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TAR-T62420-25mg25mg£254.00
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TAR-T62420-50mg50mg£369.00
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TAR-T62420-100mg100mg£550.00
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TAR-T62420-200mg200mg£752.00
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Further Information

Bioactivity:
P2Y2R/GPR17 antagonist 1 (Compound 14m) is a dual P2Y2R (IC50: 3.17 uM) and GPR17 (IC50: 1.67 uM) antagonist.
CAS:
2395016-49-4
Molecular Weight:
432.83
Pathway:
GPCR/G Protein|Endocrinology/Hormones
Purity:
0.9821
SMILES:
O=C(C1=C(Cl)C=CC=C1)NC2=CC=C(S(=O)(OC3=CC=CC([N+]([O-])=O)=C3)=O)C=C2
Target:
GPR

References

Pillaiyar T, et al. Design, synthesis and biological evaluation of suramin-derived dual antagonists of the proinflammatory G protein-coupled receptors P2Y2 and GPR17. Eur J Med Chem. 2020 Jan 15;186:111789.