TargetMol

Tetrabenazine Metabolite

Product Code:
 
TAR-T13133
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20°C
1 / 1
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CodeSizePrice
TAR-T13133-1mg1mg£227.00
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TAR-T13133-1mL1 mL * 10 mM (in DMSO)£422.00
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TAR-T13133-5mg5mg£430.00
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TAR-T13133-10mg10mg£599.00
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TAR-T13133-25mg25mg£863.00
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TAR-T13133-50mg50mg£1,179.00
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Quantity:
TAR-T13133-100mg100mg£1,589.00
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Further Information

Bioactivity:
Tetrabenazine Metabolite, a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine. Tetrabenazine Metabolite has a high affinity for VMAT2 with a Ki of 13.4 nM. Tetrabenazine Metabolite is often used to study chorea associated with Huntington's disease and other hyperactivity disorders.
CAS:
924854-60-4
Formula:
C19H29NO3
Molecular Weight:
319.44
Pathway:
Membrane transporter/Ion channel
Purity:
0.9507
SMILES:
O(C)C=1C=C2[C@@]3(N(C[C@@H](CC(C)C)[C@@H](O)C3)CCC2=CC1OC)[H]
Target:
Monoamine Transporter

References

Zhangyu Yao , et al. Preparation and evaluation of tetrabenazine enantiomers and all eight stereoisomers of dihydrotetrabenazine as VMAT2 inhibitors. Eur J Med Chem. 2011 May;46(5):1841-8.