TargetMol

GR79236

Product Code:
 
TAR-TQ0136
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
CAS:
124555-18-6
Formula:
C15H21N5O5
Molecular Weight:
351.363
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
OCC1O[C@@H](C(O)C1O)n1cnc2c(N[C@H]3CCCC3O)ncnc12
Target:
Adenosine Receptor

References

Sneyd JR, et al. Multicentre evaluation of the adenosine agonist GR79236X in patients with dental pain after third molar extraction. Br J Anaesth. 2007 May;98(5):672-676. Arulmani U, et al. Lack of effect of the adenosine A1 receptor agonist, GR79236, on capsaicin-induced CGRP release in anaesthetized pigs. Cephalalgia. 2005 Nov;25(11):1082-90.