TargetMol

Dexloxiglumide

Product Code:
 
TAR-T15105
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T15105-100mg100mgEnquire
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Further Information

Bioactivity:
Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors.
CAS:
119817-90-2
Formula:
C21H30Cl2N2O5
Molecular Weight:
461.38
Purity:
0.98
SMILES:
[H][C@](CCC(O)=O)(NC(=O)c1ccc(Cl)c(Cl)c1)C(=O)N(CCCCC)CCCOC

References

1. Scarpignato C, et al. Effect of dexloxiglumide and spiroglumide, two new CCK-receptor antagonists, on gastric emptying and secretion in the rat: evaluation of their receptor selectivity in vivo. Aliment Pharmacol Ther. 1996 Jun;10(3):411-9. 2. Maselli MA, et al. CCK1 receptor antagonist, dexloxiglumide: effects on human isolated gallbladder. Potential clinical applications. Minerva Gastroenterol Dietol. 2003 Sep;49(3):211-6.