TargetMol

CGP 36742

Product Code:
 
TAR-T14938
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
CGP 36742 is a selective antagonist of the GABAB receptor that can penetrate the blood-brain barrier after peripheral administration (IC50: 32 μM). It is useful in the treatment of depression.
CAS:
123690-78-8
Formula:
C7H18NO2P
Molecular Weight:
179.2
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CCCCP(O)(=O)CCCN
Target:
GABA Receptor

References

1. Nowak G, et al. Antidepressant-like activity of CGP 36742 and CGP 51176, selective GABAB receptor antagonists, in rodents. Br J Pharmacol. 2006 Nov;149(5):581-90.