TargetMol

YIL 781

Product Code:
 
TAR-T23543
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T23543-1mg1mg£106.00
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TAR-T23543-5mg5mg£148.00
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TAR-T23543-1mL1 mL * 10 mM (in DMSO)£171.00
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TAR-T23543-10mg10mg£195.00
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TAR-T23543-25mg25mg£334.00
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Quantity:
TAR-T23543-50mg50mg£466.00
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Quantity:
TAR-T23543-100mg100mg£624.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Ghrelin receptor antagonist
CAS:
875258-85-8
Formula:
C24H28FN3O2?HCl
Molecular Weight:
445.96
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
FC1=CC=C(C=C1)OC2=CC=C3N=C(C)N(C(C3=C2)=O)C[C@@H]4CN(C(C)C)CCC4.Cl
Target:
GHSR

References

Kawamura K, et al. Developing new PET tracers to image the growth hormone secretagogue receptor 1a (GHS-R1a). Nucl Med Biol. 2017;52:49-56. Liu S, Li B, Qin B. Ghrelin protects retinal ganglion cells against rotenone via inhibiting apoptosis, restoring mitochondrial function, and activating AKT-mTOR signaling. Neuropeptides. 2018;67:63-70. Mende F, et al. Translating biased signaling in the ghrelin receptor system into differential in vivo functions. Proc Natl Acad Sci U S A. 2018;115(43):10255-10264. Sim YB, al. Ghrelin administered spinally increases the blood glucose level in mice. Peptides. 2014;54:162-165.