TargetMol

NVP-CGM097 sulfate

Product Code:
 
TAR-T12273
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12273-5mg5mg£246.00
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TAR-T12273-50mg50mg£1,187.00
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Quantity:
TAR-T12273-100mg100mg£1,669.00
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This product comes from: United States.
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Further Information

Bioactivity:
NVP-CGM097 sulfate is a potent and selective inhibitor of MDM2 (hMDM2, IC50 of 1.7?0.1 nM).
CAS:
1313367-56-4
Formula:
C38H49ClN4O8S
Molecular Weight:
757.34
Purity:
0.98
SMILES:
OS(O)(=O)=O.COc1cc2CC(=O)N([C@@H](c3ccc(Cl)cc3)c2cc1OC(C)C)c1ccc(cc1)N(C)C[C@H]1CC[C@@H](CC1)N1CCN(C)C(=O)C1

References

1. Holzer P, et al. Discovery of a Dihydroisoquinolinone Derivative (NVP-CGM097): A Highly Potent and Selective MDM2 Inhibitor Undergoing Phase 1 Clinical Trials in p53wt Tumors. J Med Chem. 2015 Aug 27;58(16):6348-58.