TargetMol

Mavoglurant

Product Code:
 
TAR-T11951L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11951L-5mg5mg£351.00
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TAR-T11951L-50mg50mg£1,267.00
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Quantity:
TAR-T11951L-100mg100mg£1,669.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Mavoglurant is a structurally novel, non-competitive mGlu5 receptor antagonist. It has an IC50 of 30 nM in a functional assay with human mGluR5.
CAS:
543906-09-8
Formula:
C19H23NO3
Molecular Weight:
313.397
Purity:
0.98
SMILES:
[H][C@@]12CCC[C@@](O)(C#Cc3cccc(C)c3)[C@]1([H])CCN2C(=O)OC

References

1. Vranesic I, et al. AFQ056/mavoglurant, a novel clinically effective mGluR5 antagonist: identification, SAR and pharmacological characterization. Bioorg Med Chem. 2014 Nov 1;22(21):5790-5803.