TargetMol

L-368,899 hydrochloride

Product Code:
 
TAR-T11794
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T11794-50mg50mg£695.00
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TAR-T11794-100mg100mg£1,066.00
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Further Information

Bioactivity:
L-368,899 hydrochloride, used as a tocolytic agent, is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor, respectively.
CAS:
160312-62-9
Formula:
C26H43ClN4O5S2
Molecular Weight:
591.22
Purity:
0.98
SMILES:
Cl.[H][C@@]12CC[C@](CS(=O)(=O)N3CCN(CC3)c3ccccc3C)(C(C1)NC(=O)[C@H](N)CCS(C)(=O)=O)C2(C)C

References

1. Williams PD, et al. 1-((7,7-Dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo [2.2.1]-heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperaz ine (L-368,899): an orally bioavailable, non-peptide oxytocin antagonist with potential utility for managing preterm labor. J Med Chem. 1994 Mar 4;37(5):565-71.