TargetMol

GSK598809

Product Code:
 
TAR-T11496
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11496-5mg5mg£304.00
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Quantity:
TAR-T11496-50mg50mg£1,163.00
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Quantity:
TAR-T11496-100mg100mg£1,830.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
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Further Information

Bioactivity:
GSK598809 is a selective and potent dopamine D3 Receptor (DRD3) antagonist (pKi: 8.9).
CAS:
863680-45-9
Formula:
C22H23F4N5OS
Molecular Weight:
481.51
Purity:
0.98
SMILES:
Cc1ncoc1-c1nnc(SCCCN2CC3CC3(C2)c2ccc(cc2F)C(F)(F)F)n1C

References

1. Appel NM, et al. Dopamine D3 Receptor Antagonist (GSK598809) Potentiates the Hypertensive Effects of Cocaine in Conscious, Freely-Moving Dogs. J Pharmacol Exp Ther. 2015 Sep;354(3):484-92. 2. Micheli F, et al. 1,2,4-Triazolyl azabicyclo[3.1.0]hexanes: a new series of potent and selective dopamine D(3) receptor antagonists. J Med Chem. 2010 Jan 14;53(1):374-91.