TargetMol

Dopamine D2 receptor antagonist-1

Product Code:
 
TAR-T11077
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11077-1mg1mg£124.00
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TAR-T11077-2mg2mg£148.00
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TAR-T11077-5mg5mg£201.00
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TAR-T11077-1mL1 mL * 10 mM (in DMSO)£213.00
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TAR-T11077-10mg10mg£269.00
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Quantity:
TAR-T11077-25mg25mg£429.00
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Quantity:
TAR-T11077-50mg50mg£599.00
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Quantity:
TAR-T11077-100mg100mg£824.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
Dopamine D2 receptor antagonist-1 is a negative allosteric modulator (NAM) of dopamine D2 receptor (D2R), with sub-mM affinity.
CAS:
1055411-77-2
Formula:
C14H17N3S
Molecular Weight:
259.37
Purity:
0.9977
SMILES:
N=1C=NC(NC2CCC2)=C3C1SC4=C3CCCC4

References

1. Fyfe TJ, et al. Subtle modifications to a thieno[2,3-d]pyrimidine scaffold yield negative allosteric modulators and agonists of the dopamine D2 receptor. Eur J Med Chem. 2019 Apr 15;168:474-490.