TargetMol

AHR antagonist 2

Product Code:
 
TAR-T10269
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10269-1mg1mg£138.00
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TAR-T10269-5mg5mg£229.00
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TAR-T10269-1mL1 mL * 10 mM (in DMSO)£252.00
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TAR-T10269-10mg10mg£334.00
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TAR-T10269-25mg25mg£519.00
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TAR-T10269-50mg50mg£703.00
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TAR-T10269-100mg100mg£970.00
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TAR-T10269-500mg500mg£1,862.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AHR antagonist 2 is a potent aryl hydrocarbon receptor (AHR) antagonist, extracted from patent WO2019101641A1, compound example 1 (IC50s: 0.885 and 2.03 nM for human and mouse AhR).
CAS:
2338747-54-7
Formula:
C20H17F3N4O3
Molecular Weight:
418.376
Pathway:
Immunology/Inflammation
Purity:
0.98
SMILES:
C[C@@H](CO)NC(=O)c1cc(nc(n1)-c1cccnc1)-c1ccc(OC(F)(F)F)cc1
Target:
Aryl Hydrocarbon Receptor

References

1. Julien LEFRANC, et al. 2-hetarylpyrimidine-4-carboxamides as aryl hydrocarbon receptor anatgonists. WO2019101641A1.