TargetMol

Casein Kinase inhibitor A86

Product Code:
 
TAR-T39482
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T39482-25mg25mg£970.00
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Further Information

Bioactivity:
Casein Kinase inhibitor A86 is a potent and orally active casein kinase 1α (CK1α) inhibitor. Casein Kinase inhibitor A86 also inhibits of CDK7 (TFIIH) and CDK9 (P-TEFb) . Casein Kinase inhibitor A861 induces leukemia cell apoptosis , and has potent anti-leukemic activities.
CAS:
2079069-01-3
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Waleed Minzel, et al. Small Molecules Co-targeting CKI? and the Transcriptional Kinases CDK7/9 Control AML in Preclinical Models. Cell. 2018 Sep 20;175(1):171-185.e25.