TargetMol

RBI-257 Maleate

Product Code:
 
TAR-T28505
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28505-5mg5mg£850.00
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TAR-T28505-50mg50mg£1,661.00
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Quantity:
TAR-T28505-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.
CAS:
911378-38-6
Formula:
C25H32IN3O5
Molecular Weight:
581.451
Purity:
0.98
SMILES:
OC(=O)C=C/C(O)=O.CC(C)Oc1cccnc1N(C)C1CCN(Cc2ccc(I)cc2)CC1

References

1. Kula NS, Baldessarini RJ, Kebabian JW, Bakthavachalam V, Xu L. RBI-257: a highly potent dopamine D4 receptor-selective ligand. Eur J Pharmacol. 1997 Jul 23;331(2-3):333-6. PubMed PMID: 9274997. 2. Cummings DF, Ericksen SS, Schetz JA. Three amino acids in the D2 dopamine receptor regulate selective ligand function and affinity. J Neurochem. 2009 Jul;110(1):45-57. doi: 10.1111/j.1471-4159.2009.06103.x. Epub 2009 Apr 16. PubMed PMID: 19486266; PubMed Central PMCID: PMC4896224. 3. Kula NS, Tarazi FI, Baldessarini RJ, Xu L, Bakthavachalam V, Pounds S, True CD. Neuropharmacological assessment of potential dopamine D4 receptor-selective radioligands. Eur J Pharmacol. 1999 Feb 12;367(1):139-42. PubMed PMID: 10082277. 4. Saito O, Ando Y, Kusano E, Asano Y. Functional characterization of basolateral and luminal dopamine receptors in rabbit CCD. Am J Physiol Renal Physiol. 2001 Jul;281(1):F114-22. PubMed PMID: 11399652.