TargetMol

BI 689648

Product Code:
 
TAR-T14664
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14664-5mg5mg£270.00
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TAR-T14664-50mg50mg£1,099.00
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Quantity:
TAR-T14664-100mg100mg£1,629.00
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This product comes from: United States.
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Further Information

Bioactivity:
BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).
CAS:
1633009-87-6
Formula:
C16H18N4O2
Molecular Weight:
298.346
Purity:
0.98
SMILES:
COCc1cncc(c1)-c1cnc2N(CCCc2c1)C(N)=O

References

1. Weldon SM, et al. Selectivity of BI 689648, a Novel, Highly Selective Aldosterone Synthase Inhibitor: Comparison with FAD286 and LCI699 in Nonhuman Primates. J Pharmacol Exp Ther. 2016 Oct;359(1):142-50.