TargetMol

SSTR5 antagonist 1

Product Code:
 
TAR-T13005
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13005-5mg5mg£303.00
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TAR-T13005-50mg50mg£1,163.00
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Quantity:
TAR-T13005-100mg100mg£1,564.00
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Further Information

Bioactivity:
SSTR5 antagonist 1 is a selective, and orally available antagonist of somatostatin receptor subtype 5 (SSTR5)(IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively).
CAS:
1628741-91-2
Formula:
C28H34FN3O5
Molecular Weight:
511.594
Purity:
0.98
SMILES:
CCOc1cc(CN2CC3(C2)CC(=NO3)N2CCC(CC2)C(O)=O)cc(OCC)c1-c1ccc(F)cc1

References

1. Hirose H, et al. Discovery of novel 5-oxa-2,6-diazaspiro[3.4]oct-6-ene derivatives as potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonists for treatment of type 2 diabetes mellitus. Bioorg Med Chem. 2017 Aug 1;25(15):4175-4193.