TargetMol

JH295

Product Code:
 
TAR-T38710
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38710-10mg10mg£604.00
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Quantity:
TAR-T38710-25mg25mg£1,099.00
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Quantity:
TAR-T38710-50mg50mg£1,629.00
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Quantity:
TAR-T38710-100mg100mg£2,336.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
JH295 is a potent, irreversible and selective NIMA-related kinase 2 (Nek2) inhibitor with an IC 50 of 770 nM. JH295 inhibits cellular Nek2 via alkylation of Cys22. JH295 is inactive against the mitotic kinases, Cdk1, Aurora B or Plk1, and does not perturb bipolar spindle assembly or the spindle assembly checkpoint.
CAS:
1311143-71-1
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Jeffrey C Henise, et al. Irreversible Nek2 kinase inhibitors with cellular activity. J Med Chem. 2011 Jun 23;54(12):4133-46.