TargetMol

CCG-232601

Product Code:
 
TAR-T26967
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T26967-5mg5mg£850.00
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Quantity:
TAR-T26967-50mg50mg£1,661.00
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Quantity:
TAR-T26967-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CCG-232601 is a inhibitor of the Rho/MRTF/SRF transcriptional pathway.
CAS:
1922099-21-5
Formula:
C24H20ClF2N3O2
Molecular Weight:
455.89
Purity:
0.98
SMILES:
FC1(F)CC(CN(C1)C(=O)c1cccc(c1)-c1ccncc1)C(=O)Nc1ccc(Cl)cc1

References

1. Pharmacokinetic optimitzation of CCG-203971: Novel inhibitors of the Rho/MRTF/SRF transcriptional pathway as potential antifibrotic therapeutics for systemic scleroderma In Press, Corrected Proof, Available online 10 March 2017 Kim M. Hutchings, Erika M. Lisabeth, Walajapet Rajeswaran, Michael W. Wilson, Roderick J. Sorenson, Phillip L. Campbell, Jeffrey H. Ruth, Asif Amin, Pei-Suen Tsou, Jeffrey R. Leipprandt, Samuel R. Olson, Bo Wen, Ting Zhao, Duxin Sun, Dinesh Khanna, David A. Fox, Richard R. Neubig, Scott D. Larsen