TargetMol

PD-118057

Product Code:
 
TAR-T16444
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T16444-1mg1mg£197.00
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Quantity:
TAR-T16444-1mL1 mL * 10 mM (in DMSO)£341.00
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TAR-T16444-5mg5mg£389.00
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TAR-T16444-10mg10mg£544.00
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TAR-T16444-25mg25mg£830.00
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Quantity:
TAR-T16444-50mg50mg£1,099.00
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Quantity:
TAR-T16444-100mg100mg£1,460.00
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Quantity:
TAR-T16444-500mg500mg£2,850.00
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Further Information

Bioactivity:
PD-118057 is a human ether-a-go-go-related gene channel activator. It does not induce hERG blockade.
CAS:
313674-97-4
Formula:
C21H17Cl2NO2
Molecular Weight:
386.27
Pathway:
JAK/STAT signaling|Angiogenesis|Tyrosine Kinase/Adaptors|Membrane transporter/Ion channel
Purity:
0.98
SMILES:
OC(=O)c1ccccc1Nc1ccc(CCc2ccc(Cl)c(Cl)c2)cc1
Target:
HER|Potassium Channel

References

1. Mao H, et al. Pharmacologic Approach to Defective Protein Trafficking in the E637K-hERG Mutant with PD-118057 and Thapsigargin. PLoS One. 2013 Jun 19;8(6):e65481.