TargetMol

JYL 1421

Product Code:
 
TAR-T15634
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15634-50mg50mg£871.00
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Quantity:
TAR-T15634-100mg100mg£1,332.00
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This product comes from: United States.
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Further Information

Bioactivity:
JYL 1421 is an antagonist of TRPV1 receptor (IC50 = 8 nM).
CAS:
401907-26-4
Formula:
C20H26FN3O2S2
Molecular Weight:
423.57
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CC(C)(C)c1ccc(CNC(=S)NCc2ccc(NS(C)(=O)=O)c(F)c2)cc1
Target:
TRP/TRPV Channel

References

1. Jakab B, et al. Pharmacological characterization of the TRPV1 receptor antagonist JYL1421 (SC0030) in vitro and in vivo in the rat. Eur J Pharmacol. 2005 Jul 4;517(1-2):35-44.