TargetMol

KI696

Product Code:
 
TAR-T11758L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11758L-1mg1mg£195.00
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TAR-T11758L-5mg5mg£462.00
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TAR-T11758L-1mL1 mL * 10 mM (in DMSO)£547.00
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TAR-T11758L-10mg10mg£646.00
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TAR-T11758L-25mg25mg£970.00
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TAR-T11758L-50mg50mg£1,259.00
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TAR-T11758L-100mg100mg£1,661.00
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This product comes from: United States.
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Further Information

Bioactivity:
KI696 is an effective and selective inhibitor of KEAP1/NRF2 interaction. KI696 is a high-affinity probe that disrupts the Keap1/NRF2 interaction.
CAS:
1799974-70-1
Formula:
C28H30N4O6S
Molecular Weight:
550.63
Pathway:
Immunology/Inflammation
Purity:
0.98
SMILES:
COc1cc(cc2nnn(C)c12)[C@@H](CC(O)=O)c1ccc(C)c(CN2C[C@@H](C)Oc3ccccc3S2(=O)=O)c1
Target:
Nrf2

References

1. Davies TG, et al. Monoacidic Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2-Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction with High Cell Potency Identified by Fragment-Based Discovery. J Med Chem. 2016 Apr 28;59(8):3991-4006.