TargetMol

GSK-2793660

Product Code:
 
TAR-T11466
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11466-5mg5mg£483.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T11466-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T11466-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK-2793660 is an oral and irreversible inhibitor of Cathepsin C (CTSC). It can be used for the research of bronchiectasis.
CAS:
1613458-70-0
Formula:
C20H27N3O3
Molecular Weight:
357.454
Purity:
0.98
SMILES:
CC[C@H](NC(=O)C1(N)CCOCC1)C=CC(=O)N1CCc2ccccc12

References

1. Szcze?niak P, et al. The Synthesis of ?,?-Disubstituted ?-Amino Acids via Ichikawa Rearrangement. J Org Chem. 2016 Feb 5;81(3):1057-74. 2. Miller BE, et al. Epithelial desquamation observed in a phase I study of an oral cathepsin C inhibitor (GSK2793660). Br J Clin Pharmacol. 2017 Dec;83(12):2813-2820.