TargetMol

AR453588

Product Code:
 
TAR-T10362
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10362-5mg5mg£390.00
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Quantity:
TAR-T10362-50mg50mg£1,797.00
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Quantity:
TAR-T10362-100mg100mg£2,801.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AR453588 is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
CAS:
1065609-00-8
Formula:
C25H25N7O2S2
Molecular Weight:
519.64
Purity:
0.98
SMILES:
CC(=O)N1CCC(CC1)c1nsc(Nc2ncc(Sc3ccccn3)cc2Oc2cccnc2C)n1

References

1. Hinklin RJ, et al. Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator. Bioorg Med Chem. 2020 Jan 1;28(1):115232.