TargetMol

Stressin I

Product Code:
 
TAR-TP2125
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TP2125-5mg5mg£969.00
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Further Information

Bioactivity:
Potent and selective corticotropin releasing factor receptor-1 (CRF1) agonist (Ki values are 1.5 and 224 nM for CRF1 and CRF2 receptors respectively). Increases ACTH levels and increases faecal pellet output in vivo following i.p. administration.
CAS:
TP2125
Formula:
C203H337N57O56
Molecular Weight:
4472.24
Purity:
0.98
SMILES:
0

References

Rivier et al (2007) Stressin1-A, a potent cortico. releasing factor receptor 1 (CRF1)-selective peptide agonist. J.Med.Chem. 50 1668 PMID: Rivier et al (2002) Receptor-selective cortico. releasing factor analogs. Endocrin.Soc.Abstr. P2-50 Bruchas et al (2009) CRF1-R activation of the dynorphin/kappa opioid system in the mouse basolateral amygdala mediates anxiety-like behavior. PLoS One. 4 e8528 PMID: