TargetMol

Taltirelin

Product Code:
 
TAR-T7590
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7590-5mg5mg£111.00
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TAR-T7590-1mL1 mL * 10 mM (in DMSO)£113.00
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TAR-T7590-10mg10mg£136.00
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TAR-T7590-50mg50mg£324.00
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TAR-T7590-100mg100mg£526.00
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This product comes from: United States.
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Further Information

Bioactivity:
Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release))[1].
CAS:
103300-74-9
Formula:
C17H23N7O5
Molecular Weight:
405.415
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
CN1C(=O)C[C@H](NC1=O)C(=O)N[C@@H](Cc1cnc[nH]1)C(=O)N1CCC[C@H]1C(N)=O
Target:
Thyroid hormone receptor(THR)

References

Dougherty J P , Wolff B S , Cullen M J , et al. Taltirelin alleviates fatigue-like behavior in mouse models of cancer-related fatigue.[J]. Pharmacological Research, 2017, 124:1-8. Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.