TargetMol

MJN110

Product Code:
 
TAR-T5815
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T5815-5mg5mg£105.00
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TAR-T5815-1mL1 mL * 10 mM (in DMSO)£109.00
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TAR-T5815-10mg10mg£134.00
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TAR-T5815-25mg25mg£213.00
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TAR-T5815-50mg50mg£302.00
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TAR-T5815-100mg100mg£487.00
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This product comes from: United States.
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Further Information

Bioactivity:
Cravatt Reagent is a potent and selective MAGL inhibitor. Cravatt Reagent inhibits MAGL (IC50 = 9.1 nM). MJN110 Produces Opioid-Sparing Effects in a Mouse Neuropathic Pain Model.
CAS:
1438416-21-7
Formula:
C22H21Cl2N3O4
Molecular Weight:
462.33
Pathway:
Metabolism
Purity:
0.98
SMILES:
Clc1ccc(cc1)C(N1CCN(CC1)C(=O)ON1C(=O)CCC1=O)c1ccc(Cl)cc1
Target:
Lipase

References

Wilkerson J L , Niphakis M J , Grim T W , et al. The selective monoacylglycerol lipase inhibitor MJN110 produces opioid sparing effects in a mouse neuropathic pain model[J]. Journal of Pharmacology and Experimental Therapeutics, 2016:jpet.115.229971.