TargetMol

D3-βArr

Product Code:
 
TAR-T5383
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5383-5mg5mg£115.00
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Quantity:
TAR-T5383-1mL1 mL * 10 mM (in DMSO)£119.00
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TAR-T5383-10mg10mg£148.00
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TAR-T5383-25mg25mg£228.00
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TAR-T5383-50mg50mg£364.00
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Quantity:
TAR-T5383-100mg100mg£518.00
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Further Information

Bioactivity:
D3-βArr is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct TSHR activation.
CAS:
662164-09-2
Formula:
C20H23N5
Molecular Weight:
333.439
Pathway:
GPCR/G Protein
Purity:
0.9943
SMILES:
CC(Nc1nc(nc2ccccc12)N1CCNCC1)c1ccccc1
Target:
TSH Receptor

References

Neumann S, et al. Discovery of a Positive Allosteric Modulator of the Thyrotropin Receptor: Potentiation of Thyrotropin-Mediated Preosteoblast Differentiation In Vitro. J Pharmacol Exp Ther. 2018 Jan;364(1):38-45.