TargetMol

LIT927

Product Code:
 
TAR-T5207
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5207-1mg1mg£97.00
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TAR-T5207-2mg2mg£107.00
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TAR-T5207-5mg5mg£127.00
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TAR-T5207-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T5207-10mg10mg£160.00
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TAR-T5207-25mg25mg£244.00
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TAR-T5207-50mg50mg£349.00
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TAR-T5207-100mg100mg£538.00
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TAR-T5207-500mg500mg£1,091.00
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Further Information

Bioactivity:
LIT-927 is an orally active CXCL12 neutraligand (Ki: 267 nM for CXCL12 binding to CXCR4).
CAS:
2172879-52-4
Formula:
C17H13ClN2O3
Molecular Weight:
328.75
Pathway:
Autophagy; Immunology/Inflammation; GPCR/G Protein
Purity:
0.9973
SMILES:
COc1cc(ccc1O)-c1cc(nc(=O)[nH]1)-c1ccc(Cl)cc1
Target:
CXCR

References

Regenass P, et al. Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia. J Med Chem. 2018 Sep 13;61(17):7671-7686.