TargetMol

DS45500853

Product Code:
 
TAR-T40349
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
DS45500853 is an estrogen-related receptor α ( ERRα ) agonist. DS45500853 inhibits the binding between receptor-interacting protein 140 (RIP140) corepressor peptide (10 nM) and GST-ERRα ligand-binding domain (LBD; 1.2 μM) with an IC 50 value of 0.80 μM. DS45500853 can be used for the research of metabolic disorders, including type 2 diabetes mellitus (T2DM).
CAS:
2735803-28-6
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Shinozuka T, et al. Discovery of a Novel Class of ERR? Agonists. ACS Med Chem Lett. 2021 Apr 21;12(5):817-821.