TargetMol

GLUT inhibitor-1

Product Code:
 
TAR-T40083
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T40083-100mg100mgEnquire
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TAR-T40083-5mg5mg£591.00
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TAR-T40083-10mg10mg£871.00
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TAR-T40083-25mg25mg£1,669.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GLUT inhibitor-1 is an orally active GLUT inhibitor with IC50 s of 242 nM and 179 nM for GLUT1 and GLUT3. GLUT inhibitor-1 can be used in studies about cancers and autoimmune diseases.
CAS:
2421141-40-2
Formula:
C32H35N7O2
Molecular Weight:
549.67
Pathway:
Metabolism
Purity:
0.9735
SMILES:
O=C(NC1(C)CC1)COC2=CC=CC(=C2)C=3N=C(NC=4C=CC(=CC4)C=5C=NNC5)C6=C(N3)CCN(C6)C7CCC7
Target:
transporter

References

Liu KG, et al. Discovery and Optimization of Glucose Uptake Inhibitors. J Med Chem. 2020;63(10):5201-5211.