TargetMol

SR-1277

Product Code:
 
TAR-T38927
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38927-5mg5mg£850.00
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Further Information

Bioactivity:
SR-1277 is a potent, selective and ATP competitive CK1δ/ε inhibitor, with IC 50 s of 49 nM and 260 nM, respectively. SR-1277 also inhibits FLT3 , CDK4/cyclin D1 , CDK6/cyclin D3 and CDK9/cyclin K , with IC 50 s of 305 nM, 1340 nM, 311 nM and 109 nM, respectively. SR-1277 can be used for the research of cancer.
CAS:
1446715-47-4
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Bibian M, et, al. Development of highly selective casein kinase 1?/1? (CK1?/?) inhibitors with potent antiproliferative properties. Bioorg Med Chem Lett. 2013 Aug 1;23(15):4374-80.