TargetMol

GYKI-47261 dihydrochloride

Product Code:
 
TAR-T38601
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38601-5mg5mg£850.00
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Further Information

Bioactivity:
GYKI-47261 dihydrochloride is a competitive, orally active, and selective AMPA receptor antagonist with an IC 50 of 2.5 μM. GYKI-47261 has broad spectrum anticonvulsive activity and neuroprotective effects. GYKI-47261 dihydrochloride is also a potent inducer of CYP2E1.
CAS:
1217049-32-5
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Abrah?m G, et al. New non competitive AMPA antagonists. Bioorg Med Chem. 2000;8(8):2127-2143. Tam?si V, et al. GYKI-47261, a new AMPA [2-amino-3-(3-hydroxymethylisoxazole-4-yl)propionic acid] antagonist, is a CYP2E1 inducer. Drug Metab Dispos. 2003;31(11):1310-1314.