TargetMol

LDN-0088050

Product Code:
 
TAR-T37614
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T37614-5mg5mg£850.00
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Quantity:
TAR-T37614-50mg50mg£1,661.00
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Quantity:
TAR-T37614-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
LDN 0088050 is selectivity adipocyte fatty acid binding protein (AFABP, FABP4) inhibitor with Ki values of 0.29 and 1.3 μM for FABP4 and FABP3, respectively. LDN 0088050 binds to FABP4 with a Kd of 2.05 μM[1]. Ki: 0.29 μM (FABP4), 1.3 μM (FABP3)[1]Kd: 2.05 μM (FABP4)[1]
CAS:
353484-30-7
Formula:
C19H18BrNO2
Molecular Weight:
372.26
Purity:
0.98
SMILES:
OC(C(C1C2C=CC1)N3CC4C(C=CC4)C5=CC(Br)=CC2=C35)=O

References

Zhou Y, et al. The discovery of novel and selective fatty acid binding protein 4 inhibitors by virtual screening and biological evaluation. Bioorg Med Chem. 2016 Sep 15;24(18):4310-4317.