TargetMol

Epelsiban besylate

Product Code:
 
TAR-T31647
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T31647-5mg5mg£1,171.00
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TAR-T31647-50mg50mg£2,303.00
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Quantity:
TAR-T31647-100mg100mg£3,042.00
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This product comes from: United States.
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Further Information

Bioactivity:
Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.
CAS:
1159097-48-9
Formula:
C36H44N4O7S
Molecular Weight:
676.83
Purity:
0.98
SMILES:
OS(=O)(=O)c1ccccc1.CC[C@H](C)[C@H]1N([C@@H](C(=O)N2CCOCC2)c2ccc(C)nc2C)C(=O)[C@H](NC1=O)C1Cc2ccccc2C1

References

1. Mahar KM, Stier B, Fries M, McCallum SW. A single- and multiple-dose study to investigate the pharmacokinetics of epelsiban and its metabolite, GSK2395448, in healthy female volunteers. Clin Pharmacol Drug Dev. 2015 Nov;4(6):418-26. doi: 10.1002/cpdd.210. Epub 2015 Aug 26. PubMed PMID: 27137713. 2. Shinghal R, Barnes A, Mahar KM, Stier B, Giancaterino L, Condreay LD, Black L, McCallum SW. Safety and efficacy of epelsiban in the treatment of men with premature ejaculation: a randomized, double-blind, placebo-controlled, fixed-dose study. J Sex Med. 2013 Oct;10(10):2506-17. doi: 10.1111/jsm.12272. Epub 2013 Aug 12. PubMed PMID: 23937679.